{"id":53685,"date":"2025-08-15T05:40:29","date_gmt":"2025-08-15T05:40:29","guid":{"rendered":"https:\/\/rechemco.to\/?post_type=product&p=53685"},"modified":"2026-06-16T02:30:39","modified_gmt":"2026-06-16T02:30:39","slug":"fluoprazolam-cn","status":"publish","type":"product","link":"https:\/\/rechemco.to\/nl\/fluoprazolam-cn\/","title":{"rendered":"Fluoprazolam Freebase CN Export \u2013 Groothandel"},"content":{"rendered":"\n

Fluoprazolam \u2013 Piperazinyl-Substituted Benzimidazodiazepine<\/strong><\/p>\n\n\n\n

\n\n\n\n

\ud83e\uddec Overview<\/strong><\/h3>\n\n\n\n

Fluoprazolam<\/strong> is a potent synthetic benzimidazo[1,2-a][1,4]diazepine<\/strong> derivative, structurally distinct from both alprazolam and flualprazolam. It incorporates:<\/p>\n\n\n\n

    \n
  • A 2-fluorophenyl<\/strong> substitution<\/li>\n\n\n\n
  • An 8-nitro group<\/strong> on the benzimidazo core<\/li>\n\n\n\n
  • A 4-methylpiperazin-1-ylmethylene<\/strong> moiety at position 2<\/li>\n<\/ul>\n\n\n\n

    This unique substitution pattern is designed to modulate GABA<sub>A<\/sub> receptor affinity<\/strong> while altering physicochemical properties such as lipophilicity, CNS penetration, and metabolic stability.<\/p>\n\n\n\n

    \n\n\n\n

    \u269b\ufe0f Chemical Identity<\/strong><\/h3>\n\n\n\n
      \n
    • IUPAC Name<\/strong>: (Z)-6-(2-fluorophenyl)-2-((4-methylpiperazin-1-yl)methylene)-8-nitro-4H-benzo[f]imidazo[1,2-a][1,4]diazepin-1-one<\/em><\/li>\n\n\n\n
    • Molecular Formula<\/strong>: C\u2082\u2082H\u2082\u2081FN\u2086O\u2083<\/li>\n\n\n\n
    • Molecular Weight<\/strong>: ~448.46 g\/mol<\/li>\n\n\n\n
    • Chemical Class<\/strong>: Benzimidazo[1,2-a][1,4]diazepine (nitro-substituted)<\/li>\n<\/ul>\n\n\n\n
      \n\n\n\n

      \u2699\ufe0f Pharmacology<\/strong><\/h3>\n\n\n\n

      As a benzodiazepine-class ligand, Fluoprazolam is presumed to act as a positive allosteric modulator<\/strong> at the GABA<sub>A<\/sub> receptor benzodiazepine site<\/strong>. Binding enhances the effect of endogenous GABA, increasing neuronal chloride influx, leading to:<\/p>\n\n\n\n

        \n
      • Sedative-hypnotic effects<\/li>\n\n\n\n
      • Anxiolysis<\/li>\n\n\n\n
      • Anticonvulsant activity<\/li>\n\n\n\n
      • Muscle relaxation<\/li>\n<\/ul>\n\n\n\n

        The piperazinylmethylene<\/strong> side chain may alter receptor subtype selectivity or confer additional pharmacokinetic changes (e.g., slower metabolism).
        The nitro<\/strong> group in benzodiazepine analogs is often associated with longer half-life and high receptor affinity.<\/p>\n\n\n\n

        \n\n\n\n

        \ud83d\udcc8 Pharmacokinetics<\/strong> (based on class data, specific studies on Fluoprazolam limited)<\/em><\/h3>\n\n\n\n
          \n
        • Onset<\/strong>: Likely within 30\u201360 minutes (oral)<\/li>\n\n\n\n
        • Duration<\/strong>: Estimated 8\u201314 hours (possible residual sedation)<\/li>\n\n\n\n
        • Metabolism<\/strong>: Hepatic, probable CYP3A4 involvement<\/li>\n\n\n\n
        • Excretion<\/strong>: Urinary metabolites after oxidative and reductive transformations<\/li>\n<\/ul>\n\n\n\n
          \n\n\n\n

          \u26a0\ufe0f Effects & Risks<\/strong><\/h3>\n\n\n\n

          Potential desired effects<\/strong> (at controlled research doses):<\/p>\n\n\n\n

            \n
          • Profound sedation<\/li>\n\n\n\n
          • Reduced anxiety<\/li>\n\n\n\n
          • Anticonvulsant action<\/li>\n\n\n\n
          • Sleep induction<\/li>\n<\/ul>\n\n\n\n

            Adverse effects \/ overdose symptoms<\/strong>:<\/p>\n\n\n\n

              \n
            • Respiratory depression<\/li>\n\n\n\n
            • Severe motor incoordination<\/li>\n\n\n\n
            • Memory blackouts<\/li>\n\n\n\n
            • Hypotension<\/li>\n\n\n\n
            • Prolonged unconsciousness<\/li>\n<\/ul>\n\n\n\n

              Given the likely high potency, sub-milligram active quantities<\/strong> are plausible, requiring extreme caution in measurement and handling.<\/p>\n\n\n\n

              \n\n\n\n

              \u2757 Harm Reduction for Laboratory Use<\/strong><\/h3>\n\n\n\n
                \n
              • Always weigh with 0.1 mg analytical balances<\/strong> or use volumetric dilution<\/strong><\/li>\n\n\n\n
              • Avoid inhalation\/dermal exposure \u2014 use PPE and fume hood<\/li>\n\n\n\n
              • Store securely to prevent unauthorized access<\/li>\n\n\n\n
              • Keep away from heat, light, and moisture<\/li>\n<\/ul>\n\n\n\n
                \n\n\n\n

                \ud83d\udd2c Research Applications<\/strong><\/h3>\n\n\n\n

                Fluoprazolam\u2019s unusual piperazinylmethylene<\/strong> substitution makes it a valuable reference for:<\/p>\n\n\n\n

                  \n
                • Structure\u2013activity relationship (SAR) studies within benzodiazepines<\/li>\n\n\n\n
                • Pharmacokinetic modeling of bulky side chain effects<\/li>\n\n\n\n
                • Forensic standard for analytical testing of seized samples<\/li>\n<\/ul>\n\n\n\n
                  \n\n\n\n

                  \ud83c\udf0d Legal Status<\/strong><\/h3>\n\n\n\n

                  While specific scheduling varies, most jurisdictions control nitrobenzodiazepines under psychotropic substance laws or analog provisions.
                  Researchers must confirm local legality<\/strong> before acquisition or handling.<\/p>\n\n\n\n

                  \n\n\n\n

                  \ud83d\udccc Summary<\/strong><\/h3>\n\n\n\n

                  Fluoprazolam is a high-affinity benzimidazodiazepine<\/strong> with a distinctive structure, likely potent CNS depressant effects, and long duration. Its profile makes it important in forensic toxicology<\/strong> and benzodiazepine receptor research<\/strong>, but also demands stringent safety protocols<\/strong>.<\/p>\n\n\n\n

                  \n\n\n\n

                  Why Buy Fluoprazolam<\/strong> from RECHEMCO?<\/h2>\n\n\n\n

                  \u2605 We have a long trading history in the market so you benefit from our experience.
                  \u2605 Fluoprazolam<\/strong><\/strong> was tested and verified.
                  \u2605 We accept various payment methods such as Bitcoin, the main cryptocurrencies, Credit Card via Plisio and bank wire.<\/p>\n\n\n\n

                  What you will receive when you buy\u00a0Fluoprazolam<\/strong><\/strong><\/strong><\/strong>\u00a0from RECHEMCO?<\/h3>\n\n\n\n

                  \u2022\u00a0One sealed aluminum foil bag containing highest grade\u00a0Fluoprazolam<\/strong><\/strong><\/strong>
                  \u2022\u00a0white\/yellowish powder
                  \u2022\u00a099% Purity<\/p>\n","protected":false},"excerpt":{"rendered":"

                  Fluoprazolam \u2013 Piperazinyl-Substituted Benzimidazodiazepine<\/h2>\n

                  Fluoprazolam<\/strong> is a nitro-substituted benzimidazo[1,2-a][1,4]diazepine featuring a 2-fluorophenyl group and a 4-methylpiperazinylmethylene side chain. It acts as a positive allosteric modulator at GABAA<\/sub> receptors, producing potent sedative and anxiolytic effects in research models.<\/p>\n

                    \n
                  • IUPAC: (Z)-6-(2-fluorophenyl)-2-((4-methylpiperazin-1-yl)methylene)-8-nitro-4H-benzo[f]imidazo[1,2-a][1,4]diazepin-1-one<\/li>\n
                  • High receptor affinity and prolonged duration<\/li>\n
                  • Intended for forensic and pharmacological research only<\/li>\n<\/ul>\n

                    Not for human or veterinary use. Handle with extreme caution in a controlled lab environment.<\/em><\/p>\n

                    Fluoprazolam<\/strong> is ready to be shipped in 48h-72h after the payment.<\/p>\n

                    Average delivery time: 1 month.<\/p>\n

                    All the designer drugs sold on this website are intended for research and forensic applications.<\/strong><\/p>\n

                    ATTENTION!
                    <\/b>IN CASE OF LOSS, WRONG ADDRESS OR ANY OTHER ISSUE, FOR THIS PRODUCT IS NOT ALLOWED ANY RESHIP NOR REFUND<\/p>\n

                     <\/p>\n","protected":false},"featured_media":55746,"comment_status":"open","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[15],"product_tag":[1853,1861,1855,1863,1856,1849,1846,1851,1858,1848,1850,1852,1857,1862,1845,1847,1860,1312,1859,1854],"class_list":["post-53685","product","type-product","status-publish","has-post-thumbnail","product_cat-out-of-stock","product_tag-analytical-reference-benzodiazepine","product_tag-benzimidazodiazepine","product_tag-benzodiazepine-analog","product_tag-benzodiazepine-analog-toxicology","product_tag-benzodiazepine-metabolism-studies","product_tag-benzodiazepine-pharmacology","product_tag-benzodiazepine-potency-study","product_tag-benzodiazepine-receptor-binding-study","product_tag-benzodiazepine-sar-research","product_tag-cns-depressant-reference","product_tag-diazepine-research-compound","product_tag-fluoprazolam","product_tag-forensic-benzodiazepine-standard","product_tag-gaba-a-receptor-modulator","product_tag-lab-use-only-benzodiazepine","product_tag-nitro-diazepine-ligand","product_tag-nitrobenzodiazepine","product_tag-novel-benzodiazepine","product_tag-piperazinylmethylene-benzodiazepine","product_tag-sedative-hypnotic-research","first","outofstock","shipping-taxable","purchasable","product-type-variable"],"_links":{"self":[{"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/product\/53685","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/comments?post=53685"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/media\/55746"}],"wp:attachment":[{"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/media?parent=53685"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/product_brand?post=53685"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/product_cat?post=53685"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/rechemco.to\/nl\/wp-json\/wp\/v2\/product_tag?post=53685"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}